gasguide

Phenylephrine

Synthetic α1-agonist

Pure α1 agonist → vasoconstriction. No β activity.

Indications

  • Anesthesia-induced hypotension
  • OB spinal hypotension (preferred over ephedrine for fetal pH)
  • Mydriasis (ophthalmic)

Dosing

ContextAdultPediatric
Bolus50–200 mcg IV
Infusion0.15–1.5 mcg/kg/min
OB spinal prophylaxis0.5–1 mcg/kg/min infusion at spinal placement

Pharmacokinetics

Onset 1 min. Duration 10–20 min.

Hemodynamic effects

↑SVR, ↑BP. Reflex bradycardia (often ↓CO).

Side effects

  • !Bradycardia + ↓CO (relevant in poor LV function)
  • !Reduced uteroplacental flow at high dose

Contraindications

  • ×Severe LV dysfunction (relative — reduced CO with vasoconstriction)

Clinical pearls

  • OB spinal: phenylephrine maintains umbilical artery pH better than ephedrine.
  • Cardiac surgery off-pump: phenyl preferred for systemic pressure during graft anastomoses.
  • Watch for reflex bradycardia in LVH/HOCM patients.
Education only — confirm against current package inserts and institutional protocols. Doses assume normal organ function unless otherwise noted.