gasguide

Epinephrine

Adrenalin

Endogenous catecholamine, α + β agonist

α1 (vasoconstriction), α2, β1 (inotropy + chronotropy), β2 (bronchodilation, vasodilation in skeletal muscle). Dose-dependent receptor preference: low-dose β-predominant, high-dose α-predominant.

Indications

  • Anaphylaxis
  • Cardiac arrest
  • Hemodynamic support / inotropy
  • Bronchospasm
  • Local anesthetic vasoconstrictor

Dosing

ContextAdultPediatric
Anaphylaxis IM0.3–0.5 mg IM (1:1000)0.01 mg/kg IM
Anaphylaxis IV titrated10–100 mcg IV q1–2 min
Cardiac arrest1 mg IV q3–5 min0.01 mg/kg IV q3–5 min
Inotrope infusion0.02–0.5 mcg/kg/min
Local anesthetic adjunct1:200,000 (5 mcg/mL) — max 4.5 mg/kg lido + epi

Pharmacokinetics

Onset seconds. Duration 5–10 min. Catecholamine reuptake + COMT/MAO degradation.

Hemodynamic effects

↑HR, ↑contractility, ↑CO. SVR ↑ at high dose, ↓ at low dose (β2). Can paradoxically ↓BP at very low doses.

Respiratory effects

Bronchodilation. Decongestant (mucosal vasoconstriction).

Side effects

  • !Tachyarrhythmias
  • !Hyperglycemia
  • !Lactic acidosis
  • !Tissue ischemia at extravasation site (treat with phentolamine local infiltration)
  • !Pulmonary edema (high-dose, prolonged)

Contraindications

  • ×None for life-threatening indications

Clinical pearls

  • Anaphylaxis: IM lateral thigh fastest absorption; IV in resuscitation only.
  • LAST: drop epi to ≤1 mcg/kg (≤100 mcg).
  • Caution: with halothane ('sensitized myocardium' — but halothane is rarely used in 2026).
Education only — confirm against current package inserts and institutional protocols. Doses assume normal organ function unless otherwise noted.